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Discovery of new piperaquine hybrid analogs linked by triazolopyrimidine and pyrazolopyrimidine scaffolds with antiplasmodial and transmission blocking activities

Livia M. Feitosa, Rodolfo Rodrigo Florido França, Maria de Lourdes Garcia Ferreira, Anna Caroline Campos Aguiar, Guilherme Eduardo de Souza, Sarah El Chamy Maluf, Juliana Oliveira de Souza, Luana Carlos Campisano Zapata, Denise Duarte, Inês Morais, Fátima Nogueira, M. Cristina Nonato, Luiz Carlos da Silva Pinheiro, Rafael V. C. Guido, Nubia Boechat

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Pharmacology, Toxicology and Pharmaceutical Science